TargetMol

Fezagepras sodium

Product Code:
 
TAR-T12375
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T12375-1mg1mg£119.00
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TAR-T12375-5mg5mg£189.00
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TAR-T12375-1mL1 mL * 10 mM (in DMSO)£201.00
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TAR-T12375-10mg10mg£262.00
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TAR-T12375-25mg25mg£430.00
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TAR-T12375-50mg50mg£608.00
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TAR-T12375-100mg100mg£836.00
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TAR-T12375-500mg500mg£1,613.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Setogepram sodium salt is an orally active GPR40 agonist and is an antagonist or inverse agonist for GPR84, with anti-fibrotic, anti-inflammatory and anti-proliferative actions.
CAS:
1254472-97-3
Formula:
C13H17NaO2
Molecular Weight:
228.267
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.98
SMILES:
CCCCCc1cccc(CC(=O)O[Na])c1
Target:
GPR

References

1. Li Y, et al. Fatty acid receptor modulator PBI-4050 inhibits kidney fibrosis and improves glycemic control. JCI Insight. 2018 May 17;3(10). pii: 120365. 2. Grouix B, et al. PBI-4050 Reduces Stellate Cell Activation and Liver Fibrosis through Modulation of Intracellular ATP Levels and the Liver Kinase B1/AMP-Activated Protein Kinase/Mammalian Target of Rapamycin Pathway. J Pharmacol Exp Ther. 2018 Oct;367(1):71-81.