TargetMol

SUN 1334H

Product Code:
 
TAR-T13040
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
CAS:
607736-84-5
Formula:
C23H28Cl2F2N2O3
Molecular Weight:
489.38
Pathway:
GPCR/G Protein; Neuroscience; Immunology/Inflammation
Purity:
0.98
SMILES:
Cl.Cl.OC(=O)COCC=CCN1CCN(CC1)C(c1ccc(F)cc1)c1ccc(F)cc1
Target:
Histamine Receptor

References

1. Mandhane SN, et al. Preclinical efficacy and safety pharmacology of SUN-1334H, a potent orally active antihistamine agent. Drugs R D. 2008;9(2):93-112. 2. Mandhane SN, et al. Characterization of anti-inflammatory properties and evidence for no sedation liability for the novel antihistamine SUN-1334H. Int Arch Allergy Immunol. 2010;151(1):56-69.