TargetMol

ASP6432

Product Code:
 
TAR-T14335
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T14335-5mg5mg£302.00
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TAR-T14335-50mg50mg£1,163.00
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TAR-T14335-100mg100mg£1,564.00
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This product comes from: United States.
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Further Information

Bioactivity:
ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and rat LPA1, the IC50s are 11 nM and 30 nM , respectively.
CAS:
1282549-08-9
Formula:
C26H31KN4O6S2
Molecular Weight:
598.77
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
[K+].CCNS(=O)(=O)[N-]C(=O)c1csc(CN(CCCc2ccccc2)C(=O)c2cc(OC)c(C)c(OC)c2)n1
Target:
LPA Receptor

References

1. Sakamoto K, et al. Effect of ASP6432, a Novel Type 1 Lysophosphatidic Acid Receptor Antagonist, on Urethral Function and Prostate Cell Proliferation. J Pharmacol Exp Ther. 2018 Aug;366(2):390-396.