TargetMol

L-798106

Product Code:
 
TAR-T15689
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
L-798106 is a highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM). It also has micromolar activities at EP4, EP1, and EP2 receptors (Ki: 916 nM, >5000 nM, and >5000 nM at EP4, EP1, and EP2, respectively).
CAS:
244101-02-8
Formula:
C27H22BrNO4S
Molecular Weight:
536.44
Pathway:
Immunology/Inflammation; GPCR/G Protein
Purity:
0.98
SMILES:
COc1ccc(Br)cc1S(=O)(=O)NC(=O)C=Cc1ccccc1Cc1ccc2ccccc2c1
Target:
Prostaglandin Receptor

References

1. Juteau H, et al. Structure-activity relationship of cinnamic acylsulfonamide analogues on the human EP3 prostanoid receptor. Bioorg Med Chem. 2001 Aug;9(8):1977-84.