TargetMol

TRV120055

Product Code:
 
TAR-T39995
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T39995-50mg50mg£788.00
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This product comes from: United States.
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Further Information

Bioactivity:
TRV120055 is a G q -biased agonists, exhibits 10-fold larger molecular efficacies at the AT 1 R-Gq fusion protein compared with the AT 1 R-βarr2 fusion protein.
CAS:
2410957-04-7
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Rajagopal S, et, al. Quantifying ligand bias at seven-transmembrane receptors. Mol Pharmacol. 2011 Sep;80(3):367-77. Strachan RT, et, al. Divergent transducer-specific molecular efficacies generate biased agonism at a G protein-coupled receptor (GPCR). J Biol Chem. 2014 May 16; 289(20): 14211-24.