TargetMol

Naltrindole hydrochloride

Product Code:
 
TAR-T12169
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
Naltrindole hydrochloride is a highly potent and selective antagonist of non-peptide δ opioid receptor(Ki of 0.02 nM).
CAS:
111469-81-9
Formula:
C26H27ClN2O3
Molecular Weight:
450.96
Pathway:
GPCR/G Protein; Endocrinology/Hormones; Neuroscience
Purity:
0.98
SMILES:
Cl.[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC6CC6)CC[C@@]14[C@@]5(O)Cc1c2[nH]c2ccccc12)ccc3O
Target:
Opioid Receptor

References

1. Fern?ndez B, et al. Postnatal naltrindole treatments induce behavioural modifications in preweanling rats. Neurosci Lett. 2000 Mar 31;283(1):73-6. 2. Mundra JJ, et al. Naltrindole inhibits human multiple myeloma cell proliferation in vitro and in a murine xenograft model in vivo. J Pharmacol Exp Ther. 2012 Aug;342(2):273-87. 3. Chen YL, et al. Inhibition of akt/protein kinase B signaling by naltrindole in small cell lung cancer cells.