TargetMol

NCGC00249987

Product Code:
 
TAR-T12194
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
NCGC00249987 is a highly selective and allosteric Tyr phosphatase activity of inhibitor of Eya2(Eya2 ED and MBP-Eya2 FL with IC50s of 3 μM and 6.9 μM ).
CAS:
1384864-80-5
Formula:
C16H11FN4O2S
Molecular Weight:
342.35
Purity:
0.98
SMILES:
Fc1cccc(c1)C(=O)NN=Cc1ccc(Sc2ncccn2)o1

References

1. Anantharajan J, et al. Structural and Functional Analyses of an Allosteric EYA2 Phosphatase Inhibitor That Has On-Target Effects in Human Lung Cancer Cells. Mol Cancer Ther. 2019 Sep;18(9):1484-1496.