TargetMol

Norbinaltorphimine dihydrochloride

Product Code:
 
TAR-T12241
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
Norbinaltorphimine dihydrochloride is a potent and selective antagonist of κ opioid receptor.
CAS:
113158-34-2
Formula:
C40H45Cl2N3O6
Molecular Weight:
734.72
Pathway:
Neuroscience; Endocrinology/Hormones; GPCR/G Protein
Purity:
0.98
SMILES:
Cl.Cl.[H][C@@]12Oc3c4c(C[C@@]5([H])N(CC6CC6)CC[C@@]14[C@@]5(O)Cc1c4C[C@@]5(O)[C@@]6([H])Cc7ccc(O)c8O[C@@]([H])(c4[nH]c21)[C@]5(CCN6CC1CC1)c78)ccc3O
Target:
Opioid Receptor

References

1. Flax SM, et al. Effect of norbinaltorphimine on ??-tetrahydrocannabinol (THC)-induced taste avoidance in adolescent and adult Sprague-Dawley rats. Psychopharmacology (Berl). 2015 Sep;232(17):3193-201. 2. Jackson KJ, et al. Effects of the kappa opioid receptor antagonist, norbinaltorphimine, on stress and drug-induced reinstatement of nicotine-conditioned place preference in mice. Psychopharmacology (Berl). 2013 Apr;226(4):763-8.