TargetMol

Prinaberel

Product Code:
 
TAR-TQ0149
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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TAR-TQ0149-100mg100mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.
CAS:
524684-52-4
Formula:
C15H10FNO3
Molecular Weight:
271.247
Pathway:
Endocrinology/Hormones
Purity:
0.98
SMILES:
Oc1cc(C=C)c2oc(nc2c1)-c1ccc(O)c(F)c1
Target:
Estrogen/progestogen Receptor

References

Hinsche O, et al. Estrogen receptor ? selective agonists reduce invasiveness of triple-negative breast cancer cells. Int J Oncol. 2015 Feb;46(2):878-84. Xiu-li W, et al. ERB-041, a selective ER beta agonist, inhibits iNOS production in LPS-activated peritoneal macrophages of endometriosis via suppression of NF-kappaB activation. Mol Immunol. 2009 Jul;46(11-12):2413-8. Chaudhary SC, et al. Erb-041, an estrogen receptor-? agonist, inhibits skin photocarcinogenesis in SKH-1 hairless mice by downregulating the WNT signaling pathway. Cancer Prev Res (Phila). 2014 Feb;7(2):186-98.