TargetMol

L-655708

Product Code:
 
TAR-TQ0151
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
L-655708 is an effective inverse agonist of the α5 subunit-selective GABAA receptor (Ki: 0.45 nM).
CAS:
130477-52-0
Formula:
C18H19N3O4
Molecular Weight:
341.367
Pathway:
Membrane transporter/Ion channel; Neuroscience
Purity:
0.98
SMILES:
CCOC(=O)c1ncn-2c1[C@@H]1CCCN1C(=O)c1cc(OC)ccc-21
Target:
GABA Receptor

References

Saab BJ, et al. Short-term memory impairment after isoflurane in mice is prevented by the ?5 ?-aminobutyric acid type A receptorinverse agonist L-655708. Anesthesiology. 2010 Nov;113(5):1061-1071.