TargetMol

E7016

Product Code:
 
TAR-T61189
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T61189-1mg1mg£201.00
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TAR-T61189-5mg5mg£402.00
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TAR-T61189-10mg10mg£567.00
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TAR-T61189-25mg25mg£862.00
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TAR-T61189-50mg50mg£1,139.00
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Quantity:
TAR-T61189-100mg100mg£1,508.00
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This product comes from: United States.
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Further Information

Bioactivity:
E7016 is an orally available PARP inhibitor. E7016 inhibits of DNA repair. E7016 can enhance tumor cell radiosensitivity in vitro and in vivo.
CAS:
902128-92-1
Formula:
C20H19N3O3
Molecular Weight:
349.38
Pathway:
DNA Damage/DNA Repair|Chromatin/Epigenetic
Purity:
0.9816
SMILES:
O=C1NN=C2C=3C=C(C=CC3OC4=CC=CC1=C42)CN5CCC(O)CC5
Target:
PARP

References

Andrea L Russo, et al. In vitro and in vivo radiosensitization of glioblastoma cells by the poly (ADP-ribose) polymerase inhibitor E7016. Clin Cancer Res. 2009 Jan 15;15(2):607-12. W George Lai, et al. A Baeyer-Villiger oxidation specifically catalyzed by human flavin-containing monooxygenase 5. Drug Metab Dispos. 2011 Jan;39(1):61-70.