TargetMol

BRD4 Inhibitor-20

Product Code:
 
TAR-T61318
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T61318-1mg1mg£122.00
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TAR-T61318-5mg5mg£195.00
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TAR-T61318-1mL1 mL * 10 mM (in DMSO)£227.00
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TAR-T61318-10mg10mg£275.00
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TAR-T61318-25mg25mg£483.00
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TAR-T61318-50mg50mg£670.00
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Quantity:
TAR-T61318-100mg100mg£914.00
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Quantity:
TAR-T61318-500mg500mg£1,741.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
BRD4 Inhibitor-20 is a potent bromodomain protein 4 (BRD4) inhibitor with oral activity. BRD4 Inhibitor-20 has antiproliferative activity in cancer cell lines and is used in studies of various cancers, such as colon cancer.
CAS:
2490311-14-1
Molecular Weight:
358.41
Pathway:
Chromatin/Epigenetic
Purity:
1
SMILES:
O=C1NC2=CC=C(C=C2C1=C(C)C)NS(=O)(=O)C=3C=CC=CC3OC
Target:
Epigenetic Reader Domain

References

Yu Xu, et al. Design, synthesis and biological evaluation of indole-2-one derivatives as potent BRD4 inhibitors. Eur J Med Chem. 2020 Dec 15;208:112780.