TargetMol

WDR5-47

Product Code:
 
TAR-T67697
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T67697-1mg1mg£227.00
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TAR-T67697-5mg5mg£430.00
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TAR-T67697-1mL1 mL * 10 mM (in DMSO)£463.00
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TAR-T67697-10mg10mg£599.00
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TAR-T67697-25mg25mg£863.00
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TAR-T67697-50mg50mg£1,179.00
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Quantity:
TAR-T67697-100mg100mg£1,589.00
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Quantity:
TAR-T67697-500mg500mg£3,107.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
WDR5-47 is a potent small molecule to disturb the interaction of MLL1-WDR5 with IC50 value of 0.3uM.
CAS:
1422389-91-0
Molecular Weight:
406.84
Pathway:
Chromatin/Epigenetic
Purity:
0.9808
SMILES:
O=C(NC1=CC([N+]([O-])=O)=CC=C1N2CCN(C)CC2)C3=CC=C(F)C(C)=C3Cl
Target:
Histone Methyltransferase

References

Li DD, et al. Structure-based design and synthesis of small molecular inhibitors disturbing the interaction of MLL1-WDR5. Eur J Med Chem. 2016 Aug 8;118:1-8.