TargetMol

Fasudil dihydrochloride

Product Code:
 
TAR-T61382
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T61382-5mg5mg£850.00
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Quantity:
TAR-T61382-50mg50mg£1,661.00
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Quantity:
TAR-T61382-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Fasudil dihydrochloride, also known as HA-1077 and AT877, is a nonspecific inhibitor of RhoA/ROCK. It exhibits inhibitory effects on protein kinases, including ROCK1 with a Ki value of 0.33 uM, as well as ROCK2, PKA, PKC, and PKG with IC 50 values of 0.158 uM, 4.58 uM, 12.30 uM, and 1.650 uM, respectively. Additionally, Fasudil dihydrochloride demonstrates potent Ca 2+ channel blocking activity and acts as a vasodilator [1] [2] [3].
CAS:
203911-27-7
Molecular Weight:
364.29
Purity:
0.98
SMILES:
Cl.Cl.O=S(=O)(N1CCCNCC1)c1cccc2cnccc12