TargetMol

Relutrigine

Product Code:
 
TAR-T69652
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T69652-5mg5mg£930.00
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Quantity:
TAR-T69652-50mg50mg£1,821.00
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Quantity:
TAR-T69652-100mg100mg£2,319.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Relutrigine (PRAX-562) is an orally active inhibitor of persistent sodium channel . Relutrigine potently and preferentially inhibits persistent I Na induced by ATX-II (Nav 1.5 activator) or the SCN8A mutation N1768D with IC 50 values of 141 nM and 75 nM, respectively. Relutrigine exhibits potent use-dependent block and reduces neuronal intrinsic excitability. Relutrigine has effective anticonvulsant activity .
CAS:
2392951-29-8
Molecular Weight:
407.27
Purity:
0.98
SMILES:
FC=1C=C(C=NC1OCC(F)(F)F)C=2N=CC3=NN=C(N3C2)C(F)(F)OCC