TargetMol

CZS-241

Product Code:
 
TAR-T73449
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
 

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CodeSizePrice
TAR-T73449-5mg5mg£850.00
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Quantity:
TAR-T73449-50mg50mg£1,661.00
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Quantity:
TAR-T73449-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CZS-241 is an orally active and selective inhibitor of Polo-like Kinase (PLK) 4 ( IC 50 =2.6 nM). CZS-241 inhibits TRKA with an IC 50 value of 2.74 uM. CZS-241 induces apoptosis and arrests cell cycle at S/G2 phase. CZS-241 shows highly potent antiproliferative activity against leukemia cell lines, and exhibits safety against normal cell lines .
Molecular Weight:
551.98
Purity:
0.98
SMILES:
CC1=CC(=NN1)NC2=C3C=NN(C3=NC(=N2)NCC4=CC(=C(C=C4)Cl)C(=O)NC5=C(C=CC(=C5)F)F)C(C)C