TargetMol

JNJ-54717793

Product Code:
 
TAR-T9654
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T9654-10mg10mg£784.00
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Quantity:
TAR-T9654-25mg25mg£1,492.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
JNJ-54717793 is an orally active, brain penetrating, selective and high affinity orexin-1 receptor (OX1R) antagonist (plasma EC 50 =85 ng/mL). The K i values of JNJ-54717793 for hOX1R (human OX1R) and hOX2R are 16 nM and 700 nM, respectively. JNJ-54717793 is a potent compound of anxiety disorders [1] [2].
CAS:
1628843-99-1
Molecular Weight:
458.421
Purity:
0.98
SMILES:
[H][C@@]12CC[C@@]([H])([C@@H](C1)Nc1cnc(cn1)C(F)(F)F)N2C(=O)c1cccc(F)c1-c1ncccn1