TargetMol

SSTR5 antagonist 2 TFA

Product Code:
 
TAR-T13022L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T13022L-100mg100mgEnquire
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TAR-T13022L-500mg500mgEnquire
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Further Information

Bioactivity:
SSTR5 antagonist 2 TFA is a highly potent, oral active and selective antagonist of somatostatin (receptor) subtype 5 (SSTR5), with potential to treat type 2 diabetes mellitus (T2DM).
CAS:
1254733-98-6
Formula:
C34H36F4N2O7
Molecular Weight:
660.65
Purity:
0.98
SMILES:
O=C(O)C1=CC=C(C=C1)N2C(=O)CC3(C2)CCN(CC4=CC(OCC)=C(C(OCC)=C4)C=5C=CC(F)=CC5)CC3.O=C(O)C(F)(F)F

References

Liu W, et al. Discovery and Pharmacology of a Novel Somatostatin Subtype 5 (SSTR5) Antagonist: Synergy with DPP-4 Inhibition. ACS Med Chem Lett. 2018 Sep 12;9(11):1082-1087.