TargetMol

Emd 51921

Product Code:
 
TAR-T25368
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T25368-500mg500mgEnquire
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Further Information

Bioactivity:
Emd 51921 is a linear peptide renin inhibitor.
CAS:
133928-36-6
Molecular Weight:
756.974
Purity:
0.98
SMILES:
[3H]c1cccc([3H])c1CC(NC(=O)OC(C)(C)C)C(=O)NCC(=O)NC(CC1CCCCC1)C(O)CC(=O)NC(C(C)CC)C(=O)NCc1cnc(C)nc1N

References

Katz SA, Malvin RL, Lee J, Kim SH, Murray RD, Opsahl JA, Abraham PA. Analysis of active renin heterogeneity. Proc Soc Exp Biol Med. 1991 Sep;197(4):387-92. PubMed PMID: 1908097. Ziegler K, S?nger U. Binding proteins for linear renin-inhibiting peptides in basolateral plasma membranes of rat liver. Biochim Biophys Acta. 1992 Jan 31;1103(2):219-28. PubMed PMID: 1543706. Kim RB, Perry PR, Wilkinson GR. High affinity uptake by isolated rat hepatocytes of a linear pseudo-hexapeptide, ditekiren. Biochim Biophys Acta. 1997 Aug 14;1328(1):41-7. PubMed PMID: 9298943. Ziegler K, Kolac C, Ising W. ATP-dependent transport of the linear renin-inhibiting peptide EMD 51921 by canalicular plasma membrane vesicles of rat liver: evidence of drug-stimulatable ATP-hydrolysis. Biochim Biophys Acta. 1994 Dec 30;1196(2):209-17. PubMed PMID: 7841185.