TargetMol

GSK699

Product Code:
 
TAR-T32010
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T32010-100mg100mgEnquire
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TAR-T32010-500mg500mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC.
CAS:
2260944-68-9
Molecular Weight:
895.84
Purity:
0.98
SMILES:
O=C1C=2C(C(=O)N1C3C(=O)NC(=O)CC3)=CC=CC2OCCCC4=CC=C(N(CCCN(C(=O)C5=CC=C(C=C5)[C@H]6C[C@@H](NC7=C(Br)C(=O)N(C)N=C7)CN(C)C6)C)C)C=C4

References

Bassi ZI, Fillmore MC, Miah AH, Chapman TD, Maller C, Roberts EJ, Davis LC, Lewis DE, Galwey NW, Waddington KE, Parravicini V, Macmillan-Jones AL, Gongora C, Humphreys PG, Churcher I, Prinjha RK, Tough DF. Modulating PCAF/GCN5 Immune Cell Function through a PROTAC Approach. ACS Chem Biol. 2018 Oct 19;13(10):2862-2867. doi: 10.1021/acschembio.8b00705. Epub 2018 Sep 18. PubMed PMID: 30200762.