TargetMol

CHK1-IN-3

Product Code:
 
TAR-T10791
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10791-1mg1mg£227.00
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TAR-T10791-2mg2mg£306.00
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TAR-T10791-5mg5mg£430.00
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TAR-T10791-1mL1 mL * 10 mM (in DMSO)£468.00
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TAR-T10791-10mg10mg£600.00
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TAR-T10791-25mg25mg£863.00
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TAR-T10791-50mg50mg£1,179.00
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Quantity:
TAR-T10791-100mg100mg£1,589.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
CHK1-IN-3 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 0.4 nM).
CAS:
2097252-39-4
Formula:
C20H23N9O
Molecular Weight:
405.46
Pathway:
Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
N(C)C=1C(=CN=C(NC=2C=C(O[C@@H]3CCCNC3)C(C#N)=NC2)N1)C4=CN(C)N=C4
Target:
Chk

Documents

References

1. Tong L, et al. Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino)pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies. Eur J Med Chem. 2019 Jul 1;173:44-62.