TargetMol

TG4-155

Product Code:
 
TAR-T5482
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5482-1mg1mg£95.00
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TAR-T5482-2mg2mg£106.00
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TAR-T5482-5mg5mg£125.00
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TAR-T5482-1mL1 mL * 10 mM (in DMSO)£131.00
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TAR-T5482-10mg10mg£158.00
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TAR-T5482-25mg25mg£256.00
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TAR-T5482-50mg50mg£393.00
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TAR-T5482-100mg100mg£550.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
TG4-155 is a brain penetrant EP2 antagonist (KB = 2.4 nM) that is over 1000-fold less effective at EP4 (KB = 11.4 μM) and a panel of other receptors and channels
CAS:
1164462-05-8
Formula:
C23H26N2O4
Molecular Weight:
394.471
Pathway:
Immunology/Inflammation; GPCR/G Protein
Purity:
0.9914
SMILES:
COc1cc(C=CC(=O)NCCn2c(C)cc3ccccc23)cc(OC)c1OC
Target:
Prostaglandin Receptor

Documents

References

Jiang J , Dingledine R . Role of Prostaglandin Receptor EP2 in the Regulations of Cancer Cell Proliferation, Invasion, and Inflammation[J]. Journal of Pharmacology and Experimental Therapeutics, 2012, 344(2):360-367. Jiang J , Ganesh T , Du Y , et al. Small molecule antagonist reveals seizure-induced mediation of neuronal injury by prostaglandin E2 receptor subtype EP2[J]. Proceedings of the National Academy of Sciences, 2012, 109(8):3149-3154.