TargetMol

Dual FAAH/sEH-IN-1

Product Code:
 
TAR-T63536
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T63536-1mg1mg£262.00
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TAR-T63536-5mg5mg£538.00
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TAR-T63536-1mL1 mL * 10 mM (in DMSO)£644.00
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TAR-T63536-10mg10mg£692.00
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TAR-T63536-25mg25mg£1,010.00
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TAR-T63536-50mg50mg£1,332.00
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Quantity:
TAR-T63536-100mg100mg£1,765.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
Dual FAAH/sEH-IN-1 is a dual inhibitor of sEH (soluble epoxide hydrolase) (IC50: 9.6 nM) and FAAH (fatty acid amide hydrolase) (IC50: 7 nM) with high affinity and anti-inflammatory activity.
CAS:
2756099-59-7
Molecular Weight:
512.04
Pathway:
Metabolism|Neuroscience
Purity:
0.9989
SMILES:
O=C(NC1=CC=C(C=C1)C2=NC=3C=CC=CC3S2)C4CCN(CC4)S(=O)(=O)C=5C=CC=CC5Cl
Target:
FAAH|Epoxide Hydrolase

Documents

References

Wilt S, Kodani S, Valencia L, et al. Further exploration of the structure-activity relationship of dual soluble epoxide hydrolase/fatty acid amide hydrolase inhibitors. Bioorg Med Chem. 2021;51:116507.