TargetMol

NHE3-IN-3

Product Code:
 
TAR-T61480
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T61480-100mg100mgEnquire
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TAR-T61480-50mg50mgEnquire
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
NHE3-IN-3 (Compound 1) is a potent inhibitor of the isoform 3 of the Na+/H+ exchanger (NHE3). It exhibits pIC50 values of 6.2 and 6.6 against human and rat NHE3, respectively. Furthermore, NHE3-IN-3 showcases exceptional oral bioavailability of 98% in Sprague?Dawley rats [1].
CAS:
543734-50-5
Molecular Weight:
371.28
Purity:
0.98
SMILES:
CN1CC(c2cccc(c2)S(N)(=O)=O)c2cc(Cl)cc(Cl)c2C1

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